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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $28.05 | Total: $140.25 |
| 1 | 10 | $23.76 | Total: $237.60 |
| 1 | 25 | $20.13 | Total: $503.25 |
| 1 | 50 | $17.16 | Total: $858.00 |
| 1 | 100 | $14.85 | Total: $1,485.00 |
Overview
Uprosertib (GSK2141795) (GSK2141795) is a selective, ATP-competitive, and orally bioavailable Akt inhibitor with IC50 of 180 nM, 328 nM, and 38 nM for Akt 1, 2 and 3, respectively. Phase 2.
Chemical Properties
| Molecular Formula | C18H16Cl2F2N4O2 |
| Molecular Weight | 429.25 |
| CAS Numbers | 1047634-65-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cn1ncc(Cl)c1-c1cc(oc1Cl)C(=O)NC(CN)Cc1ccc(F)c(F)c1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Pachl F, et al. J Proteome Res. 2013, 12[8], 3792-3800.