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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $26.35 | Total: $131.75 |
| 1 | 10 | $22.32 | Total: $223.20 |
| 1 | 25 | $18.91 | Total: $472.75 |
| 1 | 50 | $16.12 | Total: $806.00 |
| 1 | 100 | $13.95 | Total: $1,395.00 |
Overview
Glasdegib (PF-04449913) (PF-04449913) is a potent, and orally bioavailable Smoothened (Smo) inhibitor with IC50 of 5 nM. Phase 2.
Chemical Properties
| Molecular Formula | C21H22N6O |
| Molecular Weight | 374.44 |
| CAS Numbers | 1095173-27-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN1CC[C@H](C[C@@H]1c1nc2ccccc2[nH]1)NC(=O)Nc1ccc(cc1)C#N |
Storage and Handling
0C Short Term, -20C Long Term
References
Munchhof MJ, et al. ACS Med Chem Lett. 2011, 3[2], 106-111.