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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $84.15 | Total: $420.75 |
| 1 | 10 | $71.28 | Total: $712.80 |
| 1 | 25 | $60.39 | Total: $1,509.75 |
| 1 | 50 | $51.48 | Total: $2,574.00 |
| 1 | 100 | $44.55 | Total: $4,455.00 |
Overview
Lintitript (SR 27897) is a selective CCK1 antagonist with an EC50 of 6 nM for CCK1 and 200 nM for CCK2, and a Ki value of 0.2 nM for CCK1.
Chemical Properties
| Molecular Formula | C20H14ClN3O3S |
| Molecular Weight | 411.86 |
| CAS Numbers | 136381-85-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | OC(=O)Cn1c(cc2ccccc12)C(=O)Nc1nc(cs1)-c1ccccc1Cl |
Storage and Handling
0C Short Term, -20C Long Term
References
Gully D, et al. Peripheral biological activity of SR 27897 a new potent non-peptide antagonist of CCKA receptors. Eur J Pharmacol. 1993 Feb 23;232[1] 13-9.