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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $34.85 | Total: $174.25 |
| 1 | 10 | $29.52 | Total: $295.20 |
| 1 | 25 | $25.01 | Total: $625.25 |
| 1 | 50 | $21.32 | Total: $1,066.00 |
| 1 | 100 | $18.45 | Total: $1,845.00 |
Overview
DG051 is a potent leukotriene A4 hydrolase (LTA4H) inhibitor with an IC50 of 47 nM.
Chemical Properties
| Molecular Formula | C21H25Cl2NO4 |
| Molecular Weight | 426.33 |
| CAS Numbers | 929915-58-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.OC(=O)CCCN1CCC[C@H]1COc1ccc(Oc2ccc(Cl)cc2)cc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Sandanayaka V, et al. Discovery of 4-[[2S]-2-{[4-[4-chlorophenoxy]phenoxy]methyl}-1-pyrrolidinyl]butanoic acid [DG-051] as a novel leukotriene A4 hydrolase inhibitor of leukotriene B4 biosynthesis. J Med Chem. 2010 Jan 28;53[2] 573-85.