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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $40.80 | Total: $204.00 |
| 1 | 10 | $34.56 | Total: $345.60 |
| 1 | 25 | $29.28 | Total: $732.00 |
| 1 | 50 | $24.96 | Total: $1,248.00 |
| 1 | 100 | $21.60 | Total: $2,160.00 |
Overview
Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited high affinity and selectivity for the DP1 receptor.
Chemical Properties
| Molecular Formula | C24H27N3O7S |
| Molecular Weight | 501.55 |
| CAS Numbers | 932372-01-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC(C)Oc1ccc(cc1)S(=O)(=O)N1CCN(CC1)c1ccc(-c2ncco2)c(OCC(O)=O)c1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Takahashi G, et al. Effect of the potent and selective DP1 receptor antagonist, asapiprant [S-555739], in animal models of allergic rhinitis and allergic asthma. Eur J Pharmacol. 2015 Oct 15;765 15-23.