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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $105.40 | Total: $527.00 |
| 1 | 10 | $89.28 | Total: $892.80 |
| 1 | 25 | $75.64 | Total: $1,891.00 |
| 1 | 50 | $64.48 | Total: $3,224.00 |
| 1 | 100 | $55.80 | Total: $5,580.00 |
Overview
AM103 is an effective and selective inhibitor of FLAP (IC50 = 4.2 nM).
Chemical Properties
| Molecular Formula | C36H38N3NaO4S |
| Molecular Weight | 631.76 |
| CAS Numbers | 1147872-22-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | [Na+].COc1ccc(cn1)-c1ccc(Cn2c(CC(C)(C)C([O-])=O)c(SC(C)(C)C)c3cc(OCc4ccccn4)ccc23)cc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Hutchinson JH, et al. 5-lipoxygenase-activating protein inhibitors development of 3-[3-tert-butylsulfanyl-1-[4-[6-methoxy-pyridin-3-yl]-benzyl]-5-[pyridin-2-ylmethoxy]-1H-indol-2-yl]-2,2-dimethyl-propionic acid [AM103]. J Med Chem. 2009 Oct 8;52[19] 5803-15.