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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $211.65 | Total: $1,058.25 |
| 1 | 10 | $179.28 | Total: $1,792.80 |
| 1 | 25 | $151.89 | Total: $3,797.25 |
| 1 | 50 | $129.48 | Total: $6,474.00 |
| 1 | 100 | $112.05 | Total: $11,205.00 |
Overview
CP-544439 is an orally active and potent MMP-13 inhibitor that prevents diet-induced obesity and inhibits adipogenesis in 3T3-L1 preadipocytes in mice, and can be used for the study of obesity.
Chemical Properties
| Molecular Formula | C18H19FN2O6S |
| Molecular Weight | 410.42 |
| CAS Numbers | 230954-09-3 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=C(NO)C1(NS(=O)(=O)C2=CC=C(OC3=CC=C(F)C=C3)C=C2)CCOCC1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Dalvie D, et al. Metabolism distribution and excretion of a matrix metalloproteinase-13 inhibitor, 4-[4-[4-fluorophenoxy]-benzenesulfonylamino]tetrahydropyran-4-carboxylic acid hydroxyamide [CP-544439], in rats and dogs assessment of the metabolic profile of CP-544439 in plasma and urine of humans. Drug Metab Dispos. 2008 Sep;36[9] 1869-83.