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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $31.45 | Total: $157.25 |
| 1 | 10 | $26.64 | Total: $266.40 |
| 1 | 25 | $22.57 | Total: $564.25 |
| 1 | 50 | $19.24 | Total: $962.00 |
| 1 | 100 | $16.65 | Total: $1,665.00 |
Overview
Lexibulin (CYT-997)(CYT-997) is a potent tubulin polymerization inhibitor (IC50: 10-100 nM, in Y cell lines). Lexibulin blocks the formation of the mitotic spindle and leading to cell cycle arrest at the G2M phase; this may result in disruption of the tumor vasculature and tumor blood flow, and tumor cell death.
Chemical Properties
| Molecular Formula | C24H30N6O2 |
| Molecular Weight | 434.53 |
| CAS Numbers | 917111-44-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCC[C@H](Nc1nc(ncc1C)-c1ccc(NC(=O)NCC)c(OC)c1)c1cccnc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Burns CJ, et al. Mol Cancer Ther, 2009, 8[11], 3036-3045.