Categories
- PROTAC Linker
- Protein Control Ligand
- Pathway Inhibitors
- Function Modulators
- Activators
- G Protein-Coupled Receptor Ligands
- Nuclear Receptor Ligands
- GDNF Receptors
- TNF Receptors
- Transcription Factors
- Chemokines
- Cytokine Receptors
- Biomarkers and Buffer Solutions
- Molecular Probes
- Stem Cell Research
- Alzheimer's Disease
- Apoptosis
- Cancer Research
- Epigenetics
- Metabolites
- PET/SPECT Imaging Precursors
- Customized Screening Library
- Ultra Pure Pharmacological Standard
- Tissue Microarray (TMA)
- Proteins and Antibodies
- Primary Cells
- ELISA KIT
- Natural Products
- Lab Equipments
- Humanized Mice for PDX Platform
- Rare Chemicals
- Custom Synthesis
- Antibacterial
- Antifungal
- Antioxidant
- Antiviral
- Molecular Glues
- SARS-CoV
Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $269.45 | Total: $1,347.25 |
| 1 | 10 | $228.24 | Total: $2,282.40 |
| 1 | 25 | $193.37 | Total: $4,834.25 |
| 1 | 50 | $164.84 | Total: $8,242.00 |
| 1 | 100 | $142.65 | Total: $14,265.01 |
Overview
IK-862 is a selective inhibitor of TACE (ADAM17).
Chemical Properties
| Molecular Formula | C25H27N3O4 |
| Molecular Weight | 433.5 |
| CAS Numbers | 478911-60-3 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C[C@@]1(C(=O)N([C@@H](C(NO)=O)C)CC1)C2=CC=C(OCC=3C4=C(N=C(C)C3)C=CC=C4)C=C2 |
Storage and Handling
0C Short Term, -20C Long Term
References
Georgiadis D, Yiotakis A. [2008] Specific targeting of metzincin family members with small-molecule inhibitors progress toward a multifarious challenge. Bioorg. Med. Chem., 16 [19] 8781-94. [PMID 18790648]