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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $24.65 | Total: $123.25 |
| 1 | 10 | $20.88 | Total: $208.80 |
| 1 | 25 | $17.69 | Total: $442.25 |
| 1 | 50 | $15.08 | Total: $754.00 |
| 1 | 100 | $13.05 | Total: $1,305.00 |
Overview
CK-666 is a cell-permeable inhibitor of the actin-related protein Arp23 complex, binding to and stabilizing its inactive state, thereby preventing the movement of the Arp2 and Arp3 subunits into the activated filament-like (short pitch) configuration.
Chemical Properties
| Molecular Formula | C18H17FN2O |
| Molecular Weight | 296.34 |
| CAS Numbers | 442633-00-3 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1[nH]c2ccccc2c1CCNC(=O)c1ccccc1F |
Storage and Handling
0C Short Term, -20C Long Term
References
Hetrick B, et al. Small molecules CK-666 and CK-869 inhibit actin-related protein 23 complex by blocking an activating conformational change. Chem Biol. 2013 May 23;20[5] 701-12.