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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $24.65 | Total: $123.25 |
| 1 | 10 | $20.88 | Total: $208.80 |
| 1 | 25 | $17.69 | Total: $442.25 |
| 1 | 50 | $15.08 | Total: $754.00 |
| 1 | 100 | $13.05 | Total: $1,305.00 |
Overview
MMP2-IN-2 (compound 42) is a potent and selective inhibitor of MMP-2 (matrix metalloproteinases) with an IC50 of 4.2 ?M, and it also shows inhibitory activity against MMP-13, MMP-9, and MMP-8 with IC50 values of 12, 23.3, and 25 ?M, respectively [1].
Chemical Properties
| Molecular Formula | C13H8N4O4 |
| Molecular Weight | 284.23 |
| CAS Numbers | 1772-39-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=[N+]([O-])C1=CC=C(C2=NC3=CC=C([N+]([O-])=O)C=C3N2)C=C1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Laghezza A, et al. Virtual screening identification and chemical optimization of substituted 2-arylbenzimidazoles as new non-zinc-binding MMP-2 inhibitors. Bioorg Med Chem. 2020 Feb 1;28[3] 115257.