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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $22.10 | Total: $110.50 |
| 1 | 10 | $18.72 | Total: $187.20 |
| 1 | 25 | $15.86 | Total: $396.50 |
| 1 | 50 | $13.52 | Total: $676.00 |
| 1 | 100 | $11.70 | Total: $1,170.00 |
Overview
A-317491 (ABT 202) is a non-nucleotide P2X3 ( Ki: 22 nM) and P2X23 receptor (Ki: 9 nM) antagonist, which inhibits calcium flux mediated by the receptors.
Chemical Properties
| Molecular Formula | C33H27NO8 |
| Molecular Weight | 565.57 |
| CAS Numbers | 475205-49-3 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | OC(=O)c1cc(C(O)=O)c(cc1C(O)=O)C(=O)N(Cc1cccc(Oc2ccccc2)c1)[C@H]1CCCc2ccccc12 |
Storage and Handling
0C Short Term, -20C Long Term
References
Jarvis MF,et al. A-317491, a novel potent and selective non-nucleotide antagonist of P2X3 and P2X23 receptors, reduces chronic inflammatory and neuropathic pain in the rat. Proc Natl Acad Sci U S A. 2002 Dec 24;99[26] 17179-84.