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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $26.35 | Total: $131.75 |
| 1 | 10 | $22.32 | Total: $223.20 |
| 1 | 25 | $18.91 | Total: $472.75 |
| 1 | 50 | $16.12 | Total: $806.00 |
| 1 | 100 | $13.95 | Total: $1,395.00 |
Overview
Tonapofylline is an orally active and selective antagonist of the A1 adenosine receptor (Ki: 7.4 nM for human A1). Tonapofylline can be used in studies about heart failure.
Chemical Properties
| Molecular Formula | C22H32N4O4 |
| Molecular Weight | 416.51 |
| CAS Numbers | 340021-17-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCCn1c2nc([nH]c2c(=O)n(CCC)c1=O)C12CCC(CCC(O)=O)(CC1)CC2 |
Storage and Handling
0C Short Term, -20C Long Term
References
Kiesman WF, et al. Potent and orally bioavailable 8-bicyclo[2.2.2]octylxanthines as adenosine A1 receptor antagonists. J Med Chem. 2006 Nov 30;49[24] 7119-31.