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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $170.85 | Total: $854.25 |
| 1 | 10 | $144.72 | Total: $1,447.20 |
| 1 | 25 | $122.61 | Total: $3,065.25 |
| 1 | 50 | $104.52 | Total: $5,226.00 |
| 1 | 100 | $90.45 | Total: $9,045.00 |
Overview
Novokinin acetate exhibited an affinity for the AT2 receptor with Ki of 7 nM, and its antihypertensive and vasorelaxing activities were blocked by PD123319, an AT2 receptor antagonist.
Chemical Properties
| Molecular Formula | C41H65N11O9 |
| Molecular Weight | 856.02 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC(C)C[C@@H](C(N[C@@H](CCCCN)C(N(CCC1)[C@@H]1C(N[C@@H](Cc1c[nH]c2c1cccc2)C(O)=O)=O)=O)=O)NC([C@H](CCC1)N1C([C@H](CCCNC(N)=N)N)=O)=O.CC(O)=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Masaaki Yoshikawa, et al. The pharmacological effects of novokinin; a designed peptide agonist of the angiotensin AT2 receptor. Curr Pharm Des. 2013;19[17] 3009-12.