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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $135.15 | Total: $675.75 |
| 1 | 10 | $114.48 | Total: $1,144.80 |
| 1 | 25 | $96.99 | Total: $2,424.75 |
| 1 | 50 | $82.68 | Total: $4,134.00 |
| 1 | 100 | $71.55 | Total: $7,155.00 |
Overview
MLN-4760 is an angiotensin-converting (ACE2) inhibitor(human ACE2;IC50=0.44 nM). It also has excellent selectivity (>5000-fold) versus related enzymes including human testicular ACE (IC50, >100 ?M) and bovine carboxypeptidase A (CPDA; IC50, 27 ?M).
Chemical Properties
| Molecular Formula | C19H23Cl2N3O4 |
| Molecular Weight | 428.31 |
| CAS Numbers | 305335-31-3 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC(C)C[C@H](N[C@@H](Cc1cncn1Cc1cc(Cl)cc(Cl)c1)C(O)=O)C(O)=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Dales NA, et al. Substrate-based design of the first class of angiotensin-converting enzyme-related carboxypeptidase [ACE2] inhibitors. J Am Chem Soc. 2002 Oct 9;124[40] 11852-3.