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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $62.90 | Total: $314.50 |
| 1 | 10 | $53.28 | Total: $532.80 |
| 1 | 25 | $45.14 | Total: $1,128.50 |
| 1 | 50 | $38.48 | Total: $1,924.00 |
| 1 | 100 | $33.30 | Total: $3,330.00 |
Overview
Uplarafenib (B-Raf IN 10) is a potent BRAF inhibitor with an IC50 of 50-100 nM. B-Raf IN 10 exhibits antitumor activity that may influence cell proliferation and differentiation, making it suitable for studying solid tumors.
Chemical Properties
| Molecular Formula | C22H21F3N4O4S |
| Molecular Weight | 494.49 |
| CAS Numbers | 1425485-87-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCCS(=O)(=O)Nc1cc(F)c(F)c(C(=O)c2ccc3ncc(nc3c2)N2CCOCC2)c1F |
Storage and Handling
0C Short Term, -20C Long Term
References
Yong-Liang Zhu, et al. Certain Chemical Entities, Compositions, and Methods. US20130053384 A1.