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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $141.10 | Total: $705.50 |
| 1 | 10 | $119.52 | Total: $1,195.20 |
| 1 | 25 | $101.26 | Total: $2,531.50 |
| 1 | 50 | $86.32 | Total: $4,316.00 |
| 1 | 100 | $74.70 | Total: $7,470.00 |
Overview
Bisubstrate Inhibitor 78 HCl is an NNMT inhibitor (IC50 = 1.41 ?M) with potential anticancer activity, inhibiting the proliferation of HSC-2 oral cancer cells at 100 ?M.
Chemical Properties
| Molecular Formula | C25H30ClN7O5 |
| Molecular Weight | 544 |
| CAS Numbers | 917909-71-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O[C@H]1[C@@H](O[C@@H]([C@H]1O)CN(CC[C@H](N)C(O)=O)CC2=CC3=C(C=CC=C3)C=C2)N4C5=NC=NC(N)=C5N=C4.Cl |
Storage and Handling
0C Short Term, -20C Long Term
References
Gao Y,et al. Bisubstrate Inhibitors of Nicotinamide N-Methyltransferase [NNMT] with Enhanced Activity. J Med Chem. 2019 Jul 25;62[14] 6597-6614.