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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $56.95 | Total: $284.75 |
| 1 | 10 | $48.24 | Total: $482.40 |
| 1 | 25 | $40.87 | Total: $1,021.75 |
| 1 | 50 | $34.84 | Total: $1,742.00 |
| 1 | 100 | $30.15 | Total: $3,015.00 |
Overview
FATP1-IN-1 is a potent inhibitor of fatty acid transport protein 1 (FATP1). It effectively inhibits the activity of recombinant human or mouse acyl-CoA synthetase, which is essential for the function of FATP1. The inhibition is characterized by IC50 values of 0.046 ?M for human FATP1 and 0.60 ?M for mouse FATP1.
Chemical Properties
| Molecular Formula | C18H22FN5OS |
| Molecular Weight | 375.46 |
| CAS Numbers | 1431945-95-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Fc1ccc(nc1)N1CCN(CC(=O)Nc2nc3CCCCc3s2)CC1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Matsufuji T, et al. Arylpiperazines as fatty acid transport protein 1 [FATP1] inhibitors with improved potency and pharmacokinetic properties. Bioorg Med Chem Lett. 2013;23[9] 2560-2565.