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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $29.75 | Total: $148.75 |
| 1 | 10 | $25.20 | Total: $252.00 |
| 1 | 25 | $21.35 | Total: $533.75 |
| 1 | 50 | $18.20 | Total: $910.00 |
| 1 | 100 | $15.75 | Total: $1,575.00 |
Overview
ISRIB-A15 (ISR-IN-2) is an potent inhibitor of the integrated stress response with an EC50 of 0.8 nM.
Chemical Properties
| Molecular Formula | C22H22Cl4N2O4 |
| Molecular Weight | 520.23 |
| CAS Numbers | 1628478-12-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Clc1ccc(OCC(=O)N[C@H]2CC[C@@H](CC2)NC(=O)COc2ccc(Cl)c(Cl)c2)cc1Cl |
Storage and Handling
0C Short Term, -20C Long Term
References
Hearn BR, et al. Structure-Activity Studies of Bis-O-Arylglycolamides Inhibitors of the Integrated Stress Response. ChemMedChem. 2016 Apr 19;11[8] 870-80.