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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $53.55 | Total: $267.75 |
| 1 | 10 | $45.36 | Total: $453.60 |
| 1 | 25 | $38.43 | Total: $960.75 |
| 1 | 50 | $32.76 | Total: $1,638.00 |
| 1 | 100 | $28.35 | Total: $2,835.00 |
Overview
TUG-424 significantly enhances glucose-stimulated insulin secretion at 100 nM. TUG-424 is a potent and selective free fatty acid receptor 1 agonist (EC50: 32 nM).
Chemical Properties
| Molecular Formula | C18H16O2 |
| Molecular Weight | 264.32 |
| CAS Numbers | 1082058-99-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1ccccc1C#Cc1ccc(CCC(O)=O)cc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Discovery of Potent and Selective Agonists for the Free Fatty Acid Receptor 1 [FFA1GPR40], a Potential Target for the Treatment of Type II Diabetes J. Med. Chem., 2008, 51 [22], pp 7061-7064