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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $107.10 | Total: $535.50 |
| 1 | 10 | $90.72 | Total: $907.20 |
| 1 | 25 | $76.86 | Total: $1,921.50 |
| 1 | 50 | $65.52 | Total: $3,276.00 |
| 1 | 100 | $56.70 | Total: $5,670.00 |
Overview
Mefloquine (Ro 215998), a quinoline antimalarial agent, is an anti-SARS-CoV-2 entry inhibitor. Mefloquine is also a K+ channel (KvQT1minK) antagonist with an IC50 of ~1 ?M. Mefloquine can be used for malaria, systemic lupus erythematosus, and cancer research.
Chemical Properties
| Molecular Formula | C17H16F6N2O |
| Molecular Weight | 378.31 |
| CAS Numbers | 53230-10-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(F)(F)(F)C=1C2=C(C([C@H](O)[C@]3(CCCCN3)[H])=CC(C(F)(F)F)=N2)C=CC1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Kang J, et al. Interactions of the antimalarial drug mefloquine with the human cardiac potassium channels KvLQT1minK andHERG. J Pharmacol Exp Ther. 2001 Oct;299[1] 290-6.