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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $113.05 | Total: $565.25 |
| 1 | 10 | $95.76 | Total: $957.60 |
| 1 | 25 | $81.13 | Total: $2,028.25 |
| 1 | 50 | $69.16 | Total: $3,458.00 |
| 1 | 100 | $59.85 | Total: $5,985.00 |
Overview
Chymase-IN-1 is a selective, orally active inhibitor of human mast cell chymase (IC50: 29 nM).
Chemical Properties
| Molecular Formula | C20H15ClNO4PS |
| Molecular Weight | 431.83 |
| CAS Numbers | 862090-74-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(C(NC1=CC2=C(C=C1)C=CC=C2)=O)(P(=O)(O)O)C=3C=4C(SC3)=CC=C(Cl)C4 |
Storage and Handling
0C Short Term, -20C Long Term
References
Greco MN, et al. Discovery of potent, selective, orally active, nonpeptide inhibitors of human mast cell chymase. J Med Chem. 2007 Apr 19;50[8] 1727-30.