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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $78.20 | Total: $391.00 |
| 1 | 10 | $66.24 | Total: $662.40 |
| 1 | 25 | $56.12 | Total: $1,403.00 |
| 1 | 50 | $47.84 | Total: $2,392.00 |
| 1 | 100 | $41.40 | Total: $4,140.00 |
Overview
DMT1 blocker 1 is a blocker of divalent metal transporter 1 (DMT1) with IC50 of 0.64 ?M, which is expected to block the absorption of iron by intestinal cells in vivo.
Chemical Properties
| Molecular Formula | C16H14N4O2 |
| Molecular Weight | 294.31 |
| CAS Numbers | 1354790-56-9 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1nn(c(O)c1C(=O)Nc1ccccc1)-c1ccccn1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Cadieux JA, et al. Synthesis and biological evaluation of substituted pyrazoles as blockers of divalent metal transporter 1 [DMT1]. Bioorg Med Chem Lett. 2012 Jan 1;22[1] 90-5.