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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $39.95 | Total: $199.75 |
| 1 | 10 | $33.84 | Total: $338.40 |
| 1 | 25 | $28.67 | Total: $716.75 |
| 1 | 50 | $24.44 | Total: $1,222.00 |
| 1 | 100 | $21.15 | Total: $2,115.00 |
Overview
Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity.
Chemical Properties
| Molecular Formula | C14H17N3S |
| Molecular Weight | 259.37 |
| CAS Numbers | 1055411-77-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C1CC(C1)Nc1ncnc2sc3CCCCc3c12 |
Storage and Handling
0C Short Term, -20C Long Term
References
Fyfe TJ, et al. Subtle modifications to a thieno[2,3-d]pyrimidine scaffold yield negative allosteric modulators and agonists of the dopamine D2 receptor. Eur J Med Chem. 2019 Apr 15;168 474-490.