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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $84.15 | Total: $420.75 |
| 1 | 10 | $71.28 | Total: $712.80 |
| 1 | 25 | $60.39 | Total: $1,509.75 |
| 1 | 50 | $51.48 | Total: $2,574.00 |
| 1 | 100 | $44.55 | Total: $4,455.00 |
Overview
BCAT-IN-2 is an orally active and selective inhibitor of mitochondrial branched-chain aminotransferase (BCATm), inhibits BCATm and BCATc, and is used in obesity and dyslipidemia.
Chemical Properties
| Molecular Formula | C17H14ClF2N5O |
| Molecular Weight | 377.776 |
| CAS Numbers | 1800024-45-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCCc1cc(=O)n2nc(NCc3c(F)cc(Cl)cc3F)c(C#N)c2[nH]1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Bertrand SM, et al. The Discovery of in Vivo Active Mitochondrial Branched-Chain Aminotransferase [BCATm] Inhibitors by Hybridizing Fragment and HTS Hits. J Med Chem. 2015 Sep 24;58[18] 7140-63.