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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $55.25 | Total: $276.25 |
| 1 | 10 | $46.80 | Total: $468.00 |
| 1 | 25 | $39.65 | Total: $991.25 |
| 1 | 50 | $33.80 | Total: $1,690.00 |
| 1 | 100 | $29.25 | Total: $2,925.00 |
Overview
NPAS3-IN-1 is a potent inhibitor of NPAS3-ARNT heterodimerization, modulating NPAS3 transcription by targeting the interaction between NPAS3 and ARNT at the cellular level.
Chemical Properties
| Molecular Formula | C10H5N3O2S3 |
| Molecular Weight | 295.36 |
| CAS Numbers | 2207-44-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=[N+]([O-])C1=CN=C(SC2=NC3=C(S2)C=CC=C3)S1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Li P, et al. Discovery of a highly potent NPAS3 heterodimer inhibitor by covalently modifying ARNT. Bioorg Chem. 2023 Oct;139 106676.