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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $161.50 | Total: $807.50 |
| 1 | 10 | $136.80 | Total: $1,368.00 |
| 1 | 25 | $115.90 | Total: $2,897.50 |
| 1 | 50 | $98.80 | Total: $4,940.00 |
| 1 | 100 | $85.50 | Total: $8,550.00 |
Overview
I-BET567, a potent pan-BET inhibitor with oral activity, demonstrates pIC50 values of 6.9 and 7.2 for BRD4 BD1 and BD2, respectively. This compound has exhibited efficacy in mouse models of oncology and inflammation [1].
Chemical Properties
| Molecular Formula | C17H18ClN5O2 |
| Molecular Weight | 359.81 |
| CAS Numbers | 1887237-54-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C[C@H]1C[C@@H](Nc2ncc(Cl)cn2)c2cc(ccc2N1C(C)=O)C(N)=O |
Storage and Handling
0C Short Term, -20C Long Term