Tenofovir alafenamide fumarate

Tenofovir alafenamide fumarate

AOB10559

CAS: 379270-38-9

 

Chemical Name: GS-7340 fumarate; Propan-2-yl (2S)-2-[[[(2R)-1-(6-Aminopurin-9-yl)propan-2-yl]oxymethyl-phenoxyphosphoryl]amino]propanoate fumarate

More details

1000 Items

$35.00

$35.00 per 5 mg

Quantity Discount Table - Order More To Get More Price Discount

Quantity5 mgUnit Price ($/mg or $/Unit)Final Price
15 $29.75 Total: $148.75
110 $25.20 Total: $252.00
125 $21.35 Total: $533.75
150 $18.20 Total: $910.00
1100 $15.75 Total: $1,575.00

Overview

Nucleotide reverse transcriptase inhibitor (NRTI) and a novel prodrug of the antiretroviral tenofovir

Chemical Properties

Molecular FormulaC25H33N6O9P
Molecular Weight592.55
CAS Numbers379270-38-9
SolubilityDMSO
Purity98% by HPLC
IUPAC/Chemical NamePropan-2-yl (2S)-2-[[[(2R)-1-(6-Aminopurin-9-yl)propan-2-yl]oxymethyl-phenoxyphosphoryl]amino]propanoate fumarate
SMILES CodeNC1=NC=NC2=C1N=CN2C[C@@H](C)OC[P@](OC3=CC=CC=C3)(N[C@@H](C)C(OC(C)C)=O)=O.O=C(O)/C=C/C(O)=O

Storage and Handling

0°C (short term), -20°C (long term), desiccated

Synonyms

GS-7340 fumarate

References

1) Babusis D, et al. Mechanism for effective lymphoid cell and tissue loading following oral administration of nucleotide prodrug GS-7340. Mol Pharm. 2013 Feb 4;10(2):459-66.

2) Ruane PJ, et al. Antiviral activity, safety, and pharmacokinetics/pharmacodynamics of tenofovir alafenamide as 10-day monotherapy in HIV-1-positive adults. J Acquir Immune Defic Syndr. 2013 Aug 1;63(4):449-55.