Categories
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $36.55 | Total: $182.75 |
| 1 | 10 | $30.96 | Total: $309.60 |
| 1 | 25 | $26.23 | Total: $655.75 |
| 1 | 50 | $22.36 | Total: $1,118.00 |
| 1 | 100 | $19.35 | Total: $1,935.00 |
Overview
GSK805 is a potent, orally bioavailable retinoid-related orphan receptor gamma t (ROR?t) inverse agonist that interacts with the receptor's putative ligand binding domain without exerting significant effects on DNA binding
Chemical Properties
| Molecular Formula | C23H18Cl2F3NO4S |
| Molecular Weight | 532.36 |
| CAS Numbers | 1426802-50-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Xiao S , Yosef N , Yang J , et al. Small-Molecule ROR?t Antagonists Inhibit T Helper 17 Cell Transcriptional Network by Divergent Mechanisms[J]. Immunity, 2014, 40[4] 477-489.