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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $69.70 | Total: $348.50 |
| 1 | 10 | $59.04 | Total: $590.40 |
| 1 | 25 | $50.02 | Total: $1,250.50 |
| 1 | 50 | $42.64 | Total: $2,132.00 |
| 1 | 100 | $36.90 | Total: $3,690.00 |
Overview
Sigma-LIGAND-1 is a selective Sigma Receptor ligand with IC50 values of 16 nM and 19 nM at the DTG site and the PPP site, respectively, and a Ki of 4000 nM at the dopamine D2 receptor.
Chemical Properties
| Molecular Formula | C27H33NO4 |
| Molecular Weight | 435.56 |
| CAS Numbers | 139652-01-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1c(oc2ccc(OCCCCCCN3CCC(O)CC3)cc2c1=O)-c1ccccc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Erickson RH, et al. [Aminoalkoxy]chromones. Selective sigma receptor ligands. J Med Chem. 1992 May 1;35[9] 1526-35.