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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $41.65 | Total: $208.25 |
| 1 | 10 | $35.28 | Total: $352.80 |
| 1 | 25 | $29.89 | Total: $747.25 |
| 1 | 50 | $25.48 | Total: $1,274.00 |
| 1 | 100 | $22.05 | Total: $2,205.00 |
Overview
PD 144418 oxalate is a highly potent and selective sigma 1 (?1) receptor ligand with a Ki value of 0.08 nM for ?1 and 1377 nM for ?2, exhibiting negligible affinity for other receptors, ion channels, and enzymes, and demonstrating potential antipsychotic activity.
Chemical Properties
| Molecular Formula | C20H24N2O5 |
| Molecular Weight | 372.42 |
| CAS Numbers | 1794760-28-3 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=C(O)C(=O)O.N=1OC(=CC1C=2C=CC(=CC2)C)C3=CCCN(C3)CCC |
Storage and Handling
0C Short Term, -20C Long Term
References
Akunne HC, et al. The pharmacology of the novel and selective sigma ligand, PD 144418. Neuropharmacology. 1997 Jan;36[1] 51-62.