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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $78.20 | Total: $391.00 |
| 1 | 10 | $66.24 | Total: $662.40 |
| 1 | 25 | $56.12 | Total: $1,403.00 |
| 1 | 50 | $47.84 | Total: $2,392.00 |
| 1 | 100 | $41.40 | Total: $4,140.00 |
Overview
Selisistat R-enantiomer (EX-527 (R-enantiomer)) is a SIRT1 inhibitor with much less activity than the R-enantiomer of Selisistat (IC50 of SIRT1 > 100 ?M).
Chemical Properties
| Molecular Formula | C13H13ClN2O |
| Molecular Weight | 248.71 |
| CAS Numbers | 848193-69-1 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | NC(=O)[C@@H]1CCCc2c1[nH]c1ccc(Cl)cc21 |
Storage and Handling
0C Short Term, -20C Long Term
References
Napper AD, et al. Discovery of indoles as potent and selective inhibitors of the deacetylase SIRT1. J Med Chem. 2005 Dec 15;48[25] 8045-54.