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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $36.55 | Total: $182.75 |
| 1 | 10 | $30.96 | Total: $309.60 |
| 1 | 25 | $26.23 | Total: $655.75 |
| 1 | 50 | $22.36 | Total: $1,118.00 |
| 1 | 100 | $19.35 | Total: $1,935.00 |
Overview
GLPG0974 is an antagonist of FFA2GPR43 with IC50 of 9 nM.
Chemical Properties
| Molecular Formula | C25H25ClN2O4S |
| Molecular Weight | 484.99 |
| CAS Numbers | 1391076-61-1 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C[C@@]1(CCN1C(=O)c1csc2ccccc12)C(=O)N(CCCC(O)=O)Cc1cccc(Cl)c1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Pizzonero M, et al. Discovery and optimization of an azetidine chemical series as a free fatty acid receptor 2 [FFA2] antagonist from hit to clinic. J Med Chem. 2014 Dec 11;57[23] 10044-57.