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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $106.25 | Total: $531.25 |
| 1 | 10 | $90.00 | Total: $900.00 |
| 1 | 25 | $76.25 | Total: $1,906.25 |
| 1 | 50 | $65.00 | Total: $3,250.00 |
| 1 | 100 | $56.25 | Total: $5,625.00 |
Overview
Elacestrant (RAD1901) with IC50s of 48 and 870 nM for ER? and ER?, respectively.Elacestrant
Chemical Properties
| Molecular Formula | C30H38N2O2 |
| Molecular Weight | 458.63 |
| CAS Numbers | 722533-56-4 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCNCCc1ccc(CN(CC)c2cc(OC)ccc2[C@@H]2CCc3cc(O)ccc3C2)cc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Garner F, et al. RAD1901 a novel, orally bioavailable selective estrogen receptor degrader that demonstrates antitumor activity in breast cancer xenograft models. Anticancer Drugs. 2015 Oct;26[9] 948-56.