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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $182.75 | Total: $913.75 |
| 1 | 10 | $154.80 | Total: $1,548.00 |
| 1 | 25 | $131.15 | Total: $3,278.75 |
| 1 | 50 | $111.80 | Total: $5,590.00 |
| 1 | 100 | $96.75 | Total: $9,675.00 |
Overview
CMP8 is a selective ligand for estrogen receptor. CMP8 binds to the mutant estrogen receptor ligand binding domain (ERLBD). CMP8 has IC50 values of 29 nM , 41 nM, 1100 nM and 2200 nM for MGER?, MGRER?, hER? and hER?, respectively.
Chemical Properties
| Molecular Formula | C33H34ClNO3 |
| Molecular Weight | 528.08 |
| CAS Numbers | 851107-28-3 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(C12C(C=3C(C1)=CC(O)=CC3)=C(C(=O)CC2)C4=CC=C(OCCN5CCCCC5)C=C4)C6=CC=C(Cl)C=C6 |
Storage and Handling
0C Short Term, -20C Long Term
References
Miyazaki Y, et al. Destabilizing domains derived from the human estrogen receptor. J Am Chem Soc. 2012 Mar 7;134[9] 3942-5.