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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $107.10 | Total: $535.50 |
| 1 | 10 | $90.72 | Total: $907.20 |
| 1 | 25 | $76.86 | Total: $1,921.50 |
| 1 | 50 | $65.52 | Total: $3,276.00 |
| 1 | 100 | $56.70 | Total: $5,670.00 |
Overview
Kisspeptin 234 acetate(1145998-81-7 free base) is a Kisspeptin receptor (KISS1, GPR54) antagonist; a Kisspeptin-10 analogue. It inhibits the stimulation of inositol phosphate (IP) (IC50 = 7 nM) and the release of gonadotropin-releasing hormone (GnRH) by kisspeptin-10.
Chemical Properties
| Molecular Formula | C65H82N18O15 |
| Molecular Weight | 1355.46 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(NCC(N[C@H](C(NCC(N[C@@H](C(N[C@H](C(N[C@H](C(N)=O)CC1=CC=CC=C1)=O)CCCNC(N)=N)=O)CC2=CNC3=C2C=CC=C3)=O)=O)CC4=CC=CC=C4)=O)=O)CC(N)=O)=O)CC5=CNC6=C5C=CC=C6)=O)CC(N)=O)=O)NC(C)=O.CC(O)=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Roseweir et al [2009] Discovery of potent kisspeptin antagonists delineate physiological mechanisms of gonadototrophin regulation. J.Neurosci. 29 3920 PMID