MEG hemisulfate

MEG hemisulfate

AT21967

CAS 3979-00-8

More details

1000 Items

$33.80

$33.80 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $22.10 Total: $110.50
110 $18.72 Total: $187.20
125 $15.86 Total: $396.50
150 $13.52 Total: $676.00
1100 $11.70 Total: $1,170.00

Overview

MEG hemisulfate (Mercaptoethylguanidine hemisulfate) acts as a highly potent and selective suppressor of inducible NO synthase (iNOS), demonstrating EC50 values of 11.5 ?M for iNOS, 110 ?M for ecNOS, and 60 ?M for bNOS in tissue homogenates. It is notably effective as a peroxynitrite scavenger and blocks peroxynitrite-triggered oxidative mechanisms. Furthermore, this compound offers protective benefits across various experimental inflammation prototypes, such as ischemiareperfusion injury, hemorrhagic shock, periodontitis, inflammatory bowel disease, and both endotoxic and septic shock.

Chemical Properties

Molecular FormulaC6H20N6O4S3
Molecular Weight336.44
CAS Numbers3979-00-8
SolubilityDMSO
Purity98% by HPLC
SMILES CodeO=S(O)(O)=O.N=C(NCCS)N.N=C(NCCS)N

Storage and Handling

0C Short Term, -20C Long Term

References

Southan GJ, et, al. Spontaneous rearrangement of aminoalkylisothioureas into mercaptoalkylguanidines, a novel class of nitric oxide synthase inhibitors with selectivity towards the inducible isoform. Br J Pharmacol. 1996 Feb;117[4] 619-32.