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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $60.35 | Total: $301.75 |
| 1 | 10 | $51.12 | Total: $511.20 |
| 1 | 25 | $43.31 | Total: $1,082.75 |
| 1 | 50 | $36.92 | Total: $1,846.00 |
| 1 | 100 | $31.95 | Total: $3,195.00 |
Overview
Denifanstat (FASN-IN-2) is a fatty acid synthase (FASN) inhibitor (IC50=0.052 ?M, EC50=0.072 ?M) with selective and oral activity. Denifanstat has been used in studies of steatohepatitis.
Chemical Properties
| Molecular Formula | C27H29N5O |
| Molecular Weight | 439.55 |
| CAS Numbers | 1399177-37-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1n[nH]c(n1)-c1cc(C(=O)N2CCC(CC2)c2ccc(cc2)C#N)c(C)cc1C1CCC1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Johan D., et al. Heterocyclic modulators of lipid synthesis. WO2012122391A1.