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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $32.30 | Total: $161.50 |
| 1 | 10 | $27.36 | Total: $273.60 |
| 1 | 25 | $23.18 | Total: $579.50 |
| 1 | 50 | $19.76 | Total: $988.00 |
| 1 | 100 | $17.10 | Total: $1,710.00 |
Overview
Resatorvid (TAK-242), a selective Toll-like receptor 4 (TLR4) inhibitor, binds directly to Cys747 to prevent TLR4-TIRAP interaction, thereby blocking downstream signaling. Resatorvid exhibits antitumor, anti-inflammatory, and neuroprotective activities.
Chemical Properties
| Molecular Formula | C15H17ClFNO4S |
| Molecular Weight | 361.82 |
| CAS Numbers | 243984-11-4 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCOC(=O)C1=CCCC[C@H]1S(=O)(=O)Nc1ccc(F)cc1Cl |
Storage and Handling
0C Short Term, -20C Long Term
References
Zandi Z, et al. The anticancer effect of the TLR4 inhibition using TAK-242 [resatorvid] either as a single agent or in combination with chemotherapy A novel therapeutic potential for breast cancer. J Cell Biochem. 2020 Feb;121[2] 1623-1634.