Categories
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $27.20 | Total: $136.00 |
| 1 | 10 | $23.04 | Total: $230.40 |
| 1 | 25 | $19.52 | Total: $488.00 |
| 1 | 50 | $16.64 | Total: $832.00 |
| 1 | 100 | $14.40 | Total: $1,440.00 |
Overview
GIBH-130 markedly inhibits the IL-1? secretion by activated microglia (IC50: 3.4 nM). GIBH-130 is an effective inhibitor of neuroinflammation.
Chemical Properties
| Molecular Formula | C20H20N6O |
| Molecular Weight | 360.41 |
| CAS Numbers | 1252608-59-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1cc(nnc1C(=O)N1CCN(CC1)c1ncccn1)-c1ccccc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Zhou W, Zhong G, Fu S, et al. Microglia-Based Phenotypic Screening Identifies a Novel Inhibitor of Neuroinflammation Effective in Alzheimer's Disease Models[J]. Acs Chemical Neuroscience, 2016, 7[11] 1499-1507.