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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $70.55 | Total: $352.75 |
| 1 | 10 | $59.76 | Total: $597.60 |
| 1 | 25 | $50.63 | Total: $1,265.75 |
| 1 | 50 | $43.16 | Total: $2,158.00 |
| 1 | 100 | $37.35 | Total: $3,735.00 |
Overview
DUB-IN-1, with an IC50 value of 0.24 for USP8, is an active inhibitor of ubiquitin-specific protease (USPs).
Chemical Properties
| Molecular Formula | C20H11N5O |
| Molecular Weight | 337.33 |
| CAS Numbers | 924296-18-4 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N#Cc1nc2C(=NOCc3ccccc3)c3ccccc3-c2nc1C#N |
Storage and Handling
0C Short Term, -20C Long Term
References
Colombo M, et al. Synthesis and biological evaluation of 9-oxo-9H-indeno[1,2-b]pyrazine-2,3-dicarbonitrile analogues as potential inhibitors of deubiquitinating enzymes. ChemMedChem. 2010 Apr 6;5[4] 552-8.