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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $100.30 | Total: $501.50 |
| 1 | 10 | $84.96 | Total: $849.60 |
| 1 | 25 | $71.98 | Total: $1,799.50 |
| 1 | 50 | $61.36 | Total: $3,068.00 |
| 1 | 100 | $53.10 | Total: $5,310.00 |
Overview
Dub-in-2, with an IC50 value of 0.28 for USP8, is an effective deubiquitinase inhibitor.
Chemical Properties
| Molecular Formula | C15H9N5O |
| Molecular Weight | 275.26 |
| CAS Numbers | 924296-19-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCON=C1c2ccccc2-c2nc(C#N)c(nc12)C#N |
Storage and Handling
0C Short Term, -20C Long Term
References
Colombo M, et al. Synthesis and biological evaluation of 9-oxo-9H-indeno[1,2-b]pyrazine-2,3-dicarbonitrile analogues as potential inhibitors of deubiquitinating enzymes. ChemMedChem. 2010 Apr 6;5[4] 552-8.