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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $69.70 | Total: $348.50 |
| 1 | 10 | $59.04 | Total: $590.40 |
| 1 | 25 | $50.02 | Total: $1,250.50 |
| 1 | 50 | $42.64 | Total: $2,132.00 |
| 1 | 100 | $36.90 | Total: $3,690.00 |
Overview
VLX1570 is a competitive inhibitor of proteasome DUB activity, with an IC50 ranging from 4.2 ?M to 8.6 ?M, and exhibits potent inhibition of USP14.
Chemical Properties
| Molecular Formula | C23H17F2N3O6 |
| Molecular Weight | 469.39 |
| CAS Numbers | 1431280-51-1 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | [O-][N+](=O)c1cc(C=C2CCN(CC(=Cc3ccc(F)c(c3)[N+]([O-])=O)C2=O)C(=O)C=C)ccc1F |
Storage and Handling
0C Short Term, -20C Long Term
References
Wang X et al. Synthesis and evaluation of derivatives of the proteasome deubiquitinase inhibitor b-AP15. Chem Biol Drug Des, 2015 Nov, 86[5] 1036-48.