Rokitamycin

Rokitamycin

AOB9356

CAS: 74014-51-0

 

Chemical Name: Ricamycin; Propionylleucomycin; [(2S,3S,4R,6S)-6-[(2R,3S,4R,5R,6S)-6-[[(4R,5S,6S,7R,9R,10R,11E,13E,16R)-4,10-Dihydroxy-5-methoxy-9,16-dimethyl-2-oxo-7-(2-oxoethyl)-1-oxacyclohexadeca-11,13-dien-6-yl]oxy]-4-(dimethylamino)-5-hydroxy-2-methyloxan-3-yl]oxy-2,4-dimethyl-4-propanoyloxyoxan-3-yl] butanoate

More details

1000 Items

$27.30

$27.30 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $17.85 Total: $89.25
110 $15.12 Total: $151.20
125 $12.81 Total: $320.25
150 $10.92 Total: $546.00
1100 $9.45 Total: $945.00

Overview

Macrolide antibiotic, inducing DNA fragmentation and caspase activation, resembling the progression of apoptosis, reducing the mitochondrial transmembrane potential and released cytochrome c from mitochondria to the cytosol

 

References:

https://pubmed.ncbi.nlm.nih.gov/?term=Rokitamycin+&sort=date

Chemical Properties

Molecular FormulaC42H68NO16
Molecular Weight842.99
CAS Numbers74014-51-0
SolubilityDMSO and Water
Purity98% by HPLC
IUPAC/Chemical Name3-((4R,5S,6S,7R,9R,10R,11E,13E,16R)-4-(butyryloxy)-6-(((2S,3R,4R,5S,6R)-5-(((2S,4R,5S,6S)-4,5-dihydroxy-4,6-dimethyltetrahydro-2H-pyran-2-yl)oxy)-4-(dimethylamino)-3-hydroxy-6-methyltetrahydro-2H-pyran-2-yl)oxy)-10-hydroxy-5-methoxy-9,16-dimethyl-2-oxo-7-(2-oxoethyl)oxacyclohexadeca-11,13-dien-3-yl)propanoate
InChl KeyWMPXTDMRSHZXNQ-TYEDIMFNSA-M
InChl CodeInChI=1S/C42H69NO16/c1-10-14-31(48)57-37-28(17-18-30(46)47)40(51)54-24(3)15-12-11-13-16-29(45)23(2)21-27(19-20-44)36(38(37)53-9)59-41-34(49)33(43(7)8)35(25(4)56-41)58-32-22-42(6,52)39(50)26(5)55-32/h11-13,16,20,23-29,32-39,41,45,49-50,52H,10,14-15,17-19,21-22H2,1-9H3,(H,46,47)/p-1/b12-11+,16-13+/t23-,24-,25-,26+,27+,28?,29+,32+,33-,34-,35-,36+,37-,38+,39+,41+,42-/m1/s1
SMILES CodeO[C@H]([C@@H](N(C)C)[C@@H]([C@@H](C)O1)O[C@H]2C[C@@]([C@H]([C@H](C)O2)O)(C)O)[C@@H]1O[C@@H]3[C@H](OC)[C@H](OC(CCC)=O)C(CCC([O-])=O)C(O[C@H](C)C/C=C/C=C/[C@H](O)[C@H](C)C[C@@H]3CC=O)=O

Storage and Handling

0°C (short term), -20°C (long term), desiccated

Synonyms

Rokitamycin

References

1) Kim JH, Lee YJ, Sohn HJ, Song KJ, Kwon D, Kwon MH, Im KI, Shin HJ. Therapeutic effect of rokitamycin in vitro and on experimental meningoencephalitis due to Naegleria fowleri. Int J Antimicrob Agents. 2008 Nov;32(5):411-7. doi: 10.1016/j.ijantimicag.2008.05.018. Epub 2008 Aug 30. PubMed PMID: 18762406.