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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $22.10 | Total: $110.50 |
| 1 | 10 | $18.72 | Total: $187.20 |
| 1 | 25 | $15.86 | Total: $396.50 |
| 1 | 50 | $13.52 | Total: $676.00 |
| 1 | 100 | $11.70 | Total: $1,170.00 |
Overview
Tenapanor (RDX 5791) is an inhibitor of the sodium-proton (Na(+)H(+)) exchanger NHE3, which plays a prominent role in sodium handling in the gastrointestinal tract and kidney. Tenapanor possesses an excellent preclinical safety profile and, as of now, there are no serious concerns about its side effects.
Chemical Properties
| Molecular Formula | C50H66Cl4N8O10S2 |
| Molecular Weight | 1145.05 |
| CAS Numbers | 1234423-95-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN1C[C@@H](c2cccc(c2)S(=O)(=O)NCCOCCOCCNC(=O)NCCCCNC(=O)NCCOCCOCCNS(=O)(=O)c2cccc(c2)[C@@H]2CN(C)Cc3c(Cl)cc(Cl)cc23)c2cc(Cl)cc(Cl)c2C1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Johansson SA, Knutsson M, Leonsson-Zachrisson M, Rosenbaum DP. Effect of Food Intake on the Pharmacodynamics of Tenapanor A Phase 1 Study. Clin Pharmacol Drug Dev. 2017 Mar 24. doi 10.1002cpdd.341. [Epub ahead of print] PubMed PMID 28339149.