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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $211.65 | Total: $1,058.25 |
| 1 | 10 | $179.28 | Total: $1,792.80 |
| 1 | 25 | $151.89 | Total: $3,797.25 |
| 1 | 50 | $129.48 | Total: $6,474.00 |
| 1 | 100 | $112.05 | Total: $11,205.00 |
Overview
Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic and cardiovascular activities.Besipirdine inhibits voltage-dependent sodium-potassium channels and inhibits biogenic amine uptake.Besipirdine reduces schedule-induced irritability and thirst and enhances cholinergic and adrenergic activity in the CNS in the rat. Besipirdine reduces schedule-induced thirst and enhances cholinergic and adrenergic neurotransmission in the central nervous system.
Chemical Properties
| Molecular Formula | C16H17N3 |
| Molecular Weight | 251.33 |
| CAS Numbers | 119257-34-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N=1C=CC(=CC1)N(N2C=CC=3C=CC=CC32)CCC |
Storage and Handling
0C Short Term, -20C Long Term
References
Woods-Kettelberger AT,et al. Besipirdine [HP 749] reduces schedule-induced polydipsia in rats. Brain Res Bull. 1996;41[2] 125-30.