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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $80.75 | Total: $403.75 |
| 1 | 10 | $68.40 | Total: $684.00 |
| 1 | 25 | $57.95 | Total: $1,448.75 |
| 1 | 50 | $49.40 | Total: $2,470.00 |
| 1 | 100 | $42.75 | Total: $4,275.00 |
Overview
PF-04745637 is a potent and selective TRPA1 antagonist with an IC50 of 17 nM [1].
Chemical Properties
| Molecular Formula | C27H32ClF3N2O2 |
| Molecular Weight | 509 |
| CAS Numbers | 1917294-46-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | OC1(CCN(CC1)C(CNC(=O)C1(CCCC1)c1ccc(Cl)cc1)Cc1ccccc1)C(F)(F)F |
Storage and Handling
0C Short Term, -20C Long Term
References
Laurie B. Schenkel, et al. The discovery of a potent series of carboxamide TRPA1 antagonists. J. Med. Chem. 2016, 59, 6, 2794-2809.