OMDM-5

OMDM-5

AT12306

CAS 616884-66-3

More details

1000 Items

$163.80

$163.80 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $107.10 Total: $535.50
110 $90.72 Total: $907.20
125 $76.86 Total: $1,921.50
150 $65.52 Total: $3,276.00
1100 $56.70 Total: $5,670.00

Overview

OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing weak ligand activity at cannabinoid type 1 receptor (CB1, Ki=4.9 ?M). OMDM-5 is a selective anandamide cellular uptake (ACU) inhibitor(Ki = 4.8 ?M).

Chemical Properties

Molecular FormulaC26H44N2O3
Molecular Weight432.64
CAS Numbers616884-66-3
SolubilityDMSO
Purity98% by HPLC
SMILES CodeC(NNC(CCCCCCCC=CCCCCCCCC)=O)C1=CC(OC)=C(O)C=C1

Storage and Handling

0C Short Term, -20C Long Term

References

Ortar G, et al. Novel selective and metabolically stable inhibitors of anandamide cellular uptake. Biochem Pharmacol. 2003 May 1;65[9] 1473-81.