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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $48.45 | Total: $242.25 |
| 1 | 10 | $41.04 | Total: $410.40 |
| 1 | 25 | $34.77 | Total: $869.25 |
| 1 | 50 | $29.64 | Total: $1,482.00 |
| 1 | 100 | $25.65 | Total: $2,565.00 |
Overview
Obafistat is a potent inhibitor of aldo-keto reductase AKR1C3 with an IC50 of 1.2 nM for human AKR1C3.
Chemical Properties
| Molecular Formula | C15H16FN5O3S |
| Molecular Weight | 365.38 |
| CAS Numbers | 2160582-57-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Fc1cccc(c1)S(=O)(=O)N1C2CCC1CN(C2)C(=O)c1cnn[nH]1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Marcus Koppitz, et al. [8-[phenylsulfonyl]-3,8-diazabicyclo[3.2.1]oct-3-yl] [1h-1,2,3-triazol-4-yl]methanones. WO2017202817A1.