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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $93.50 | Total: $467.50 |
| 1 | 10 | $79.20 | Total: $792.00 |
| 1 | 25 | $67.10 | Total: $1,677.50 |
| 1 | 50 | $57.20 | Total: $2,860.00 |
| 1 | 100 | $49.50 | Total: $4,950.00 |
Overview
Cis-22a is a TRPV6 inhibitor (IC50 = 0.32 ?M), which exhibits selectivity against related TRPV channels and calcium channels. cis-22a displays antiproliferative effects on T47D human breast cancer cells.
Chemical Properties
| Molecular Formula | C24H30F3N3O2 |
| Molecular Weight | 449.51 |
| CAS Numbers | 1819366-84-1 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(C(O)=O)(F)(F)F.CC=1C=C([C@H]2CC[C@H](CC2)N3CCN(CC3)C=4C=CC=NC4)C=CC1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Humer C, et al. TRPV6 Regulation by Cis-22a and Cholesterol. Biomolecules. 2022;12[6] 804.